Sacubitril Hemicalcium

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沙 库 比 曲 钙盐 Sacubitril Hemicalcium 1369773-39-6 Mu nzu
沙 库 比 曲 钠盐 149690-05-1 Mu nzu
LCZ-4 1426129-50-1 Mu nzu
LCZ-7 1012341-48-8 Mu nzu
LCZ-8 1012341-50-2 Mu nzu
LCZ-9 149690-12-0 Mu nzu

 

Amavu n'amavuko

Umunyu wa AHU-377 ni umunyu wa hemicalcium yumunyu wa AHU-377.Ni inhibitori ya neprilysin ifite IC50 agaciro ka 5 nM [1].

AHU-377 hamwe na angiotensin II AT1 reseptor antagonist valsartan bahimba LCZ696 mukigereranyo cya 1: 1.LCZ696 ni reseptor ya angiotensin neprilysin inhibitor.Irashobora kugabanya umuvuduko wamaraso kandi irashobora kuba imiti mishya yo kuvura kunanirwa k'umutima.AHU-377 ni ibiyobyabwenge, birashobora guhindurwa na enzymatique clavage ya Ethyl ester muburyo bukora LBQ657.Biravugwa ko AHU-377 (30 na 100 mg / kg, PO) ishobora gutera antivypertensique mu buryo bushingiye ku mbeba ya DAHI-SS.Ariko muri imbeba ya hypertension ya DOCA-umunyu, irerekana kugabanuka guke [2, 3].

Reba:
[1] Ksander GM, Ghai RD, deJesus R, Diefenbacher CG, Yuan A, Berry C, Sakane Y, Trapani A. Dicarboxylic aside dipeptide itabogamye ya endopeptidase.J Med Chem.1995 Gicurasi 12;38 (10): 1689-700.
[2] Amajwi AA, Dorhout B, van der Meer P. Uruhare rushoboka rwa valsartan + AHU377 (LCZ696) mukuvura kunanirwa k'umutima.Impuguke Opin Iperereza Ibiyobyabwenge.2013 Kanama; 22 (8): 1041-7.
[3] Laxminarayan G Hegde, Cecile Yu, Cheruvu Madhavi n'abandi.Kugereranya efficacy ya AHU-377, inhibitor ikomeye ya neprilysin, muburyo bubiri bwimbeba ya hypertension.Imiti ya BMC 2011, 11 (Umugereka 1): P33.

Imiterere yimiti

Sacubitril Hemicalcium

CERTIFICATE

2018 GMP-2
原料药GMP证书201811(captopril ,thalidomide etc)
GMP-of-PMDA-in-Chanyoo-平成28年08月03日 Nantong-Chanyoo-Pharmatech-Co
FDA-EIR-Letter-201901

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