Bictegravir 1611493-60-7

Ibisobanuro bigufi:

Izina rya API Kwerekana Udushya Itariki yo kurangiriraho ipatanti (Amerika)
Bictegravir 1611493-60-7 Indwara ya VIH-1 Ubumenyi bwa Galeedi Ukuboza 19, 2033


Ibisobanuro birambuye

Ibiranga ibicuruzwa

KUBONA UMUSARURO

Ibisobanuro

Bictegravir nigitabo gishya, cyanduza virusi ya VIH-1 hamwe na IC50 ya 7.5 nM.

Muri Vitro

Bictegravir (BIC) ibuza ibikorwa byo kwimura umurongo hamwe na IC50 ya 7.5± 0.3 nM.Ugereranije no kubuza ibikorwa byo kwimura imirongo, Bictegravir ninzitizi ikomeye cyane ya 3-gutunganya ibikorwa bya VIH-1 IN, hamwe na IC50 ya 241±51 nM.Bictegravir yongerera imbaraga uruziga rwa 2-LTR ~ inshuro 5 ugereranije no kugenzura urw'agashinyaguro kandi igabanya ibicuruzwa biva mu mahanga byanduye inshuro 100.Bictegravir irabuza cyane kwandura virusi ya VIH-1 muri selile MT-2 na MT-4 hamwe na EC50s ya 1.5 na 2.4 nM.Bictegravir yerekana ingaruka zikomeye za virusi muri CD4 + T ya lymphocytes na macrophage ikomoka kuri monocyte, hamwe na EC50s ya 1.5±0.3 nM na 6.6±4.1 nM, bikurikiranye nagaciro kabonetse mumirongo ya T-selile [1].

MCE ntabwo yemeje ubwigenge ubu buryo.Nibisobanuro gusa.

Umubare wa NCT Umuterankunga Imiterere Itariki yo gutangiriraho

Icyiciro

NCT03998176 Kaminuza ya Nebraska | Ubumenyi bwa Galeedi VIH-1-kwandura Ku ya 9 Ukwakira 2019

Icyiciro cya 4

NCT03789968 Kaminuza ya Thomas Jefferson | Kaminuza ya Maryland, Parike ya College | Ubuzima bwa Kaminuza ya Indiana | Ikigo cy’ibitaro bya Brooklyn | Kaminuza ya Illinois i Chicago | Nova mu majyepfo y’iburasirazuba | Kaminuza ya Californiya, San Francisco VIH + SIDA Ku ya 1 Nzeri 2019
NCT04249037 Kaminuza ya Colorado, Denver | Ubumenyi bwa Galeedi VIH + SIDA Ku ya 1 Werurwe 2020

Ntabwo ari ngombwa

NCT04132674 Ikigo cyita ku ndwara zanduza Vancouver Indwara ya Immunodeficiency Yumuntu Yanduye | Gukoresha ibiyobyabwenge Ku ya 26 Ugushyingo 2018

Icyiciro cya 4

NCT04054089 Cristina Mussini | Kaminuza ya Modena na Reggio Emilia Kwandura virusi itera SIDA Nzeri 2019

Icyiciro cya 4

NCT04155554 Azienda Ospedaliera Universitaria Senese | Kaminuza Gatolika yumutima Mutagatifu | Ospedale Policlinico San Martino | Azienda Ospedaliera San Paolo | Ospedale Amedeo di Savoia VIH-1-kwandura Ku ya 29 Mutarama 2020

Icyiciro cya 3

NCT02275065 Ubumenyi bwa Galeedi Kwandura VIH-1 Ukwakira 2014

Icyiciro cya 1

NCT03711253 Kaminuza yo mu majyepfo ya California Kwandura virusi itera SIDA Ku ya 14 Ukwakira 2019

Icyiciro cya 4

NCT02400307 Ubumenyi bwa Galeedi VIH Ku ya 17 Mata 2015

Icyiciro cya 1

NCT03499483 Ubuzima bwabaturage Kwirinda virusi itera SIDA Ku ya 24 Mutarama 2019

Icyiciro cya 4

NCT03502005 Midland Research Group, Inc. | Ubumenyi bwa Galeedi Virusi ya immunodeficiency ya muntu Ku ya 1 Werurwe 2018

Icyiciro cya 4

Imiterere yimiti

Bictegravir-1611493-60-7

CERTIFICATE

2018 GMP-2
原料药GMP证书201811(captopril ,thalidomide etc)
GMP-of-PMDA-in-Chanyoo-平成28年08月03日 Nantong-Chanyoo-Pharmatech-Co
FDA-EIR-Letter-201901

Gucunga neza

Quality management1

Icyifuzo18Imishinga yo gusuzuma ireme ryemejwe4, na6imishinga iremezwa.

Quality management2

Sisitemu mpuzamahanga yo gucunga neza ubuziranenge yashyizeho urufatiro rukomeye rwo kugurisha.

Quality management3

Igenzura ryiza rinyura mubuzima bwose bwibicuruzwa kugirango hamenyekane ingaruka nziza nubuvuzi.

Quality management4

Itsinda ryumwuga ushinzwe kugenzura ibikorwa byujuje ubuziranenge mugihe cyo gusaba no kwiyandikisha.

Gucunga UMUSARURO

cpf5
cpf6

Koreya Countec Amacupa yo gupakira

cpf7
cpf8

Tayiwani CVC Icupa ryuzuye

cpf9
cpf10

Ubutaliyani CAM Ubuyobozi bwo gupakira

cpf11

Imashini yo Kudage Fette

cpf12

Ubuyapani Viswill Tablet Detector

cpf14-1

Icyumba cyo kugenzura DCS

UMUFATANYABIKORWA

Ubufatanye mpuzamahanga
International cooperation
Ubufatanye mu ngo
Domestic cooperation

  • Mbere:
  • Ibikurikira:

  • Andika ubutumwa bwawe hano hanyuma utwohereze

    Ibyiciro byibicuruzwa